Philippe Maillos' bibliography

Recent patents & publications

  • Preparation of 15-sustituted derivatives of securinine useful in the treatment of cancer WO 2016203054
  • Preparation of securinine derivatives useful in the treatment of cancer WO 2016087596
  • Synthesis and antiproliferative and metabolic evaluations of novel securinine derivatives. ACS Medicinal Chemistry Letters(2016), 7(4), 403-407
  • Highly diastereoselective 1,6-conjugate addition of arylboronic acids to securinin. Synlett (2016), 27(7), 1077-1082
  • Synthesis and biological evaluation of new securinine analogues as potential anticancer agents. European Journal of Medicinal Chemistry (2016), 109, 287-293
  • Enantioselective synthesis of both enantiomers of mequitazine through iridium-catalysed asymmetric hydrogenation of nonfunctionalizes cyclic enamine. Synlett (2014), 25(11), 1606-1610
  • Preparation of 1-[(2,3-dihydrobenzo[1,4]dioxin-2-yl)methyl]piperidin-4-yl derivatives as partial agonists or antagonist of the D2 and D3 dopamine receptors and antagonists of adrenergic alpha2C receptors for treatment of neuropsychiatric disorders WO 2014106660